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Gridegalutamide

Chemical Structure : Gridegalutamide

CAS No.: 2446929-86-6

Gridegalutamide (BMS-986409)

Catalog No.: PC-23836Not For Human Use, Lab Use Only.

Gridegalutamide (BMS-986409) is an orally bioavailable androgen receptor (AR) degrader, with potential antineoplastic activity.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

Gridegalutamide (BMS-986409) is an orally bioavailable androgen receptor (AR) degrader, with potential antineoplastic activity.

Physicochemical Properties

M.Wt 818.92
Formula C41H45F3N8O5S
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

2-[(2R)-4-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-ethylphenoxy]ethyl]-2-methylpiperazin-1-yl]-N-[3-[[(3R)-2,6-dioxopiperidin-3-yl]amino]phenyl]acetamide

References

1. Patent WO2020132014 A1.

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