HEAL-116 | 3βHSD1 inhibitor | Probechem Biochemicals

Chemical Structure : HEAL-116

HEAL-116 (HEAL116)

Catalog No.: PC-24810Not For Human Use, Lab Use Only.

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Biological Activity

HEAL-116 is a potent, selective 3β-hydroxysteroid dehydrogenase type 1 (3βHSD1) inhibitor, shows binding specificity to the substrate-binding pocket of 3βHSD1 and effectively neutralizes the local charge environment.
HEAL-116 robustly inhibits 3βHSD1 activity and exerts pronounced antitumor effect in biochemical, cellular, and mouse models.

Physicochemical Properties

M.Wt	371.82
Formula	C20H18ClNO4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-(4-Chloro-3-(morpholinomethyl) phenyl)-7-hydroxy-4H-chromen-4-one

References

1. He D, et al. Proc Natl Acad Sci U S A. 2025 Jul;122(26):e2422267122.

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HEAL-116 (HEAL116)

Biological Activity

Physicochemical Properties

References

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