Chemical Structure : HSD-016
CAS No.:
946396-92-5
HSD-016
(HSD016, HSD 016)
Catalog No. : PC-35574Not For Human Use, Lab Use Only.
HSD-016 (HSD016) is a potent, selective, and efficacious 11β-HSD1 inhibitor with IC50 of 149 and 530 nM for mouse and human 11β-HSD1, respectively.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-3557401
Biological Activity
HSD-016 (HSD016) is a potent, selective, and efficacious 11β-HSD1 inhibitor with IC50 of 149 and 530 nM for mouse and human 11β-HSD1, respectively.
Physicochemical Properties
M.Wt
514.459
Formula
C21H21F7N2O3S
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
(R)-1,1,1-trifluoro-2-(3-((R)-4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazin-1-ylsulfonyl)phenyl)propan-2-ol
References
1. Wan ZK, et al. J Org Chem.
2. Hong SP, et al. Eur J Pharmacol.
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