You are here:Home-Chemical Inhibitors & Agonists-Cell Cycle/DNA Damage-DNA Repair Protein -HUHS-015
HUHS-015

Chemical Structure : HUHS-015

CAS No.: 1453097-13-6

HUHS-015 (HUHS015)

Catalog No.: PC-42079Not For Human Use, Lab Use Only.

HUHS-015 (HUHS015) is a potent, orally active prostate cancer antigen-1 (PCA-1/ALKBH3) inhibitor with IC50 of 0.67 uM.

Packing Price Stock Quantity
25 mg $128 In stock
50 mg $198 In stock
100 mg $348 In stock
500 mg Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

HUHS-015 (HUHS015) is a potent, orally active prostate cancer antigen-1 (PCA-1/ALKBH3) inhibitor with IC50 of 0.67 uM.
HUHS-015 significantly suppresses the growth of DU145 cells in vitro and in a mouse xenograft model.

Physicochemical Properties

M.Wt 318.3724
Formula C19H18N4O
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

DMSO: ≥ 34 mg/mL

Chemical Name/SMILES

1H-Pyrazol-5-ol, 3-methyl-1-(6-methyl-1H-benzimidazol-2-yl)-4-(phenylmethyl)-

References

1. Nakao S, et al. Bioorg Med Chem Lett. 2014 Feb 15;24(4):1071-4.

2. Mabuchi M, et al. In Vivo. 2015 Jan-Feb;29(1):39-43.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: