INCB13739 | 11β-HSD1 inhibitor | Probechem Biochemicals

Chemical Structure : INCB13739

CAS No.: 869974-19-6

INCB13739 (INCB-13739, INCB 13739)

Catalog No.: PC-27071Not For Human Use, Lab Use Only.

INCB13739 (INCB-13739) is a potent, selective 11β-hydroxysteroid dehydrogenase 1 (11β-HSD1) inhibitor with enzymatic IC50 of 3.2 nM, inhibits 11β-HSD1 in PBMCs with IC50 of 1.1 nM.

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Biological Activity

INCB13739 (INCB-13739) is a potent, selective 11β-hydroxysteroid dehydrogenase 1 (11β-HSD1) inhibitor with enzymatic IC50 of 3.2 nM, inhibits 11β-HSD1 in PBMCs with IC50 of 1.1 nM.

Physicochemical Properties

M.Wt	467.53
Formula	C28H25N3O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-N-Methyl-5-(4-(1-(3-oxo-3H-spiro[isobenzofuran-1,3'-pyrrolidine]-1'-carbonyl)cyclopropyl)phenyl)picolinamide

References

1. Zhang C, et al. Bioorg Med Chem Lett. 2022 Aug 1;69:128782.

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INCB13739 (INCB-13739, INCB 13739)

Biological Activity

Physicochemical Properties

References

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