You are here:Home-Chemical Inhibitors & Agonists-Metabolic Enzyme/Protease-11β-HSD-INCB13739
INCB13739

Chemical Structure : INCB13739

CAS No.: 872506-67-7

INCB13739 (INCB-13739;INCB 13739)

Catalog No.: PC-35575Not For Human Use, Lab Use Only.

INCB13739 (INCB-13739) is a potent, selective, oral 11βHSD1 inhibitor (IC50=1.1 nM) with high seelctivity over other dehydrogenases, glucocorticoid and mineralocorticoid receptors..

Packing Price Stock Quantity
5 mg $288 In stock
10 mg $458 In stock
25 mg $758 In stock
50 mg Get quote
100 mg Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

INCB13739 (INCB-13739) is a potent, selective, oral 11β-HSD1 inhibitor (IC50=1.1 nM) with high seelctivity over other dehydrogenases, glucocorticoid and mineralocorticoid receptors.

Physicochemical Properties

M.Wt 398.946
Formula C19H27ClN2O3S
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

(3S)-1-[(3-Chloro-2-methylphenyl)sulfonyl]-N-cyclohexyl-3-piperidinecarboxamide

References

1. Rosenstock J, et al. Diabetes Care. 2010 Jul;33(7):1516-22.

2. Ge R, et al. Curr Med Chem. 2010;17(5):412-22.

3. Anagnostis P, et al. Metabolism. 2013 Jan;62(1):21-33.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: