JJ-450 | AR inhibitor | Probechem Biochemicals

Chemical Structure : JJ-450

JJ-450 (JJ450)

Catalog No.: PC-49173Not For Human Use, Lab Use Only.

JJ-450 is a novel analogue of IMTPPE and direct and specific inhibitor of androgen receptor (AR) transcriptional activity, blocks AR recruitment to androgen-responsive elements and suppresses AR target gene expression.

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Biological Activity

JJ-450 is a novel analogue of IMTPPE and direct and specific inhibitor of androgen receptor (AR) transcriptional activity, blocks AR recruitment to androgen-responsive elements and suppresses AR target gene expression.
JJ-450 also inhibits ARv7 transcriptional activity and its target gene expression.

Physicochemical Properties

M.Wt	372.868
Formula	C21H22ClFN2O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(4-(5-chloro-2-methylphenyl)piperazin-1-yl)(2-(4-fluorophenyl)cyclopropyl)methanone

References

1. Yang Z, et al. Mol Cancer Ther. 2020 Jan;19(1):75-88.

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JJ-450 (JJ450)

Biological Activity

Physicochemical Properties

References

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