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Chemical Structure : JTC-801
CAS No.: 244218-51-7
Catalog No.: PC-62626Not For Human Use, Lab Use Only.
JTC-801 is a highly potent, selective, orally active NOP receptor (ORL1) antagonist with Ki of 8.2 nM, shows 12.5-, 129- and 1055-fold selectivity over human μ-, κ- and δ-opioid receptors respectively.
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|---|---|---|---|
| 25 mg | $98 | In stock | |
| 50 mg | $148 | In stock | |
| 100 mg | $258 | In stock | |
| 250 mg | Get quote |
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JTC-801 is a highly potent, selective, orally active NOP receptor (ORL1) antagonist with Ki of 8.2 nM, shows 12.5-, 129- and 1055-fold selectivity over human μ-, κ- and δ-opioid receptors respectively.
JTC-801 demonstrates anti-nociceptive effects in acute pain models in vivo.
| M.Wt | 447.963 | |
| Formula | C26H26ClN3O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
N-(4-Amino-2-methyl-6-quinolinyl)-2-[(4-ethylphenoxy)methyl]benzamide hydrochloride |
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1. Yamada H, et al. Br J Pharmacol, 2002, 135(2), 323-332.
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