JTT251 | PDHK inhibitor | Probechem Biochemicals

Chemical Structure : JTT251

Catalog No.: PC-24276Not For Human Use, Lab Use Only.

JTT251 (JTT-251) is a potent, selective inhibitor of pyruvate dehydrogenase kinase (PDK, PDHK), bind to the allosteric lipoamide-binding domain.

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Biological Activity

JTT251 (JTT-251) is a potent, selective inhibitor of pyruvate dehydrogenase kinase (PDK, PDHK), bind to the allosteric lipoamide-binding domain.

M.Wt	503.52
Formula	C26H28F3N3O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-2-(4-(9-hydroxy-2-(3-hydroxy-3-methylbutoxy)-9-(trifluoromethyl)-9H-fluoren-4-yl)-1H-pyrazol-1-yl)-2-methylpropanamide

1. T.S. Motomura, Gakujun, Pyrazole-amide compound and medicinal uses thereof. WO2014142290 (2014).