KGP-420 |CAS:2082762-29-4 Probechem Biochemicals

Chemical Structure : KGP-420

KGP-420 (KGP420)

Catalog No.: PC-62812Not For Human Use, Lab Use Only.

KGP-420 is the water-soluble phosphate prodrug of KGP-94 in vivo studies, KGP-94 is a potent, selective cathepsin L inhibitor with IC50 of 189 nM.

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Biological Activity

KGP-420 is the water-soluble phosphate prodrug of KGP-94 in vivo studies, KGP-94 is a potent, selective cathepsin L inhibitor with IC50 of 189 nM.
KGP-420 readily converts to KGP-94, and shows cytotoxicity against HUVECs with GI50 of 20.2 uM.

Physicochemical Properties

M.Wt	476.192
Formula	C14H13BrN3Na2O4PS
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(E)-3-((3-bromophenyl)(2-carbamothioylhydrazono)methyl)phenyl dihydrogen phosphate, disodium salt

References

1. Parker EN, et al. Bioorg Med Chem Lett. 2017 Mar 1;27(5):1304-1310.

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KGP-420 (KGP420)

Biological Activity

Physicochemical Properties

References

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