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Ketanserin tartrate

Chemical Structure : Ketanserin tartrate

CAS No.: 83846-83-7

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Ketanserin tartrate (R41468 tartrate)

Catalog No.: PC-42654Not For Human Use, Lab Use Only.

A high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

A high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C; also has a high affinity antagonist for the H1 receptor (Ki= 2 nM) and α1-adrenergic receptor (Ki=40 nM); an antihypertensive agent.

Hypertension

Approved

Physicochemical Properties

M.Wt 545.5136
Formula C26H28FN3O9
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

H2O: 30 mg/mL (Need ultrasonic and warming)
Chemical Name/SMILES

2,4(1H,3H)-Quinazolinedione, 3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-, (2R,3R)-2,3-dihydroxybutanedioate (1:1)

References

1. Creed-Carson M, et al. Behav Brain Res. 2011 Jun 1;219(2):273-9.

2. Catafau AM, et al. J Cereb Blood Flow Metab. 2010 May;30(5):985-93.

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