L-869298 (L-869,298)

Chemical Structure : L-869298

Catalog No.: PC-28125Not For Human Use, Lab Use Only.

L-869298 (L-869,298) is a potent, selective and orally active PDE4 inhibitor with IC50 of 0.5 nM for PDE4A, shows less active against hERG.

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Biological Activity

L-869298 (L-869,298) is a potent, selective and orally active PDE4 inhibitor with IC50 of 0.5 nM for PDE4A, shows less active against hERG.

M.Wt	570.45
Formula	C23H18F8N2O4S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-3-(2-(3-cyclopropoxy-4-(difluoromethoxy)phenyl)-2-(2-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)thiazol-5-yl)ethyl)pyridine 1-oxide

1. Friesen RW, et al. J Med Chem. 2003 Jun 5;46(12):2413-26.