LEI-106 | DAGL-α/ABHD6 inhibitor | Probechem Biochemicals

Chemical Structure : LEI-106

CAS No.: 1620582-23-1

LEI-106 (LEI 106)

Catalog No.: PC-20127Not For Human Use, Lab Use Only.

LEI-106 (LEI 106) is a potent, dual DAGL-α/ABHD6 inhibitor with Ki values of 0.7/0.8 uM, respectively.

Packing	Price	Stock
5 mg	$248	In stock
10 mg	$398	In stock
25 mg	$598	In stock
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Biological Activity

LEI-106 (LEI 106) is a potent, dual DAGL-α/ABHD6 inhibitor with Ki values of 0.7/0.8 uM, respectively.
LEI-106 is a sulfonamide derivative in the biochemical assay with an IC50 of 18 nM for DAGL-α and inhibited the hydrolysis of [14C]-sn-1-oleoyl-2-arachidonoyl-glycerol, the natural substrate of DAGL-α with Ki of 0.7 uM.

Physicochemical Properties

M.Wt	481.56
Formula	C26H27NO6S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-((2,2-dimethylchroman-6-yl)sulfonyl)-N-(4-phenoxybenzyl)glycine

References

1. Freek J Janssen, et al. J Med Chem. 2014 Aug 14;57(15):6610-22.

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LEI-106 (LEI 106)

Biological Activity

Physicochemical Properties

References

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