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LGD-2226

Chemical Structure : LGD-2226

CAS No.: 328947-93-9

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LGD-2226 (LGD2226)

Catalog No.: PC-35143Not For Human Use, Lab Use Only.

LGD-2226 (LGD2226) is an orally active, selective androgen receptor modulator (SARM) with binding Ki of 1 nM, >1000-fold selectivity over GR,PR, MR and ER.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    LGD-2226 (LGD2226) is an orally active, selective androgen receptor modulator (SARM) with binding Ki of 1 nM, >1000-fold selectivity over GR,PR, MR and ER.
    LGD2226 is fully active in cell-based models of bone and muscle, exhibits anabolic activity on muscle and bone with reduced impact on prostate growth in rodent models.
    LGD2226 is also efficacious in a sex-behavior model in male rats measuring mounts, intromissions, ejaculations, and copulation efficiency.

    Physicochemical Properties

    M.Wt 392.225
    Formula C14H9F9N2O
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    6-(bis-(2,2,2-trifluoroethyl)amino)-4-trifluoromethyl-1H-quinolin-2-one

    References

    1. Miner JN, et al. Endocrinology. 2007 Jan;148(1):363-73.

    2. van Oeveren A, et al. J Med Chem. 2006 Oct 19;49(21):6143-6.

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