Chemical Structure : LGD-3303
CAS No.: 917891-35-1
Catalog No.: PC-61861Not For Human Use, Lab Use Only.
LGD-3303 is an orally available, brain-penetrant nonsteroidal selective androgen receptor modulator (SARM) that that shows little or no cross-reactivity with related nuclear receptors.
Packing | Price | Stock | Quantity |
---|---|---|---|
10 mg | $128 | In stock | |
25 mg | $198 | In stock | |
50 mg | Get quote | ||
100 mg | Get quote |
Bulk size, bulk discount!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
LGD-3303 is an orally available, brain-penetrant nonsteroidal selective androgen receptor modulator (SARM) that that shows little or no cross-reactivity with related nuclear receptors.
LGD-3303 has potent activity on levator ani muscle but is a partial agonist on the preputial gland and ventral prostate in a castrated rat model of androgen deficiency。
LGD-3303 enhances male-directed sexual preference, proceptive behavior, and lordosis behavior in sexually experienced, but not sexually naive, female rats.
M.Wt | 342.743 | |
Formula | C16H14ClF3N2O | |
Appearance | Solid | |
Storage |
|
|
Solubility |
10 mM in DMSO |
|
Chemical Name/SMILES |
9-Chloro-2-ethyl-1-methyl-3-(2,2,2-trifluoroethyl)-3H-pyrrolo(3,2-F)quinolin-7(6H)-one |
1. Vajda EG, et al. J Pharmacol Exp Ther. 2009 Feb;328(2):663-70.
2. Vajda EG, et al. J Bone Miner Res. 2009 Feb;24(2):231-40.
3. Kudwa AE, et al. Endocrinology. 2010 Jun;151(6):2659-68.
Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright