Chemical Structure : LGD-6972
CAS No.:
1207989-09-0
LGD-6972
(LGD6972, RVT1502)
Catalog No. : PC-43093Not For Human Use, Lab Use Only.
LGD-6972 (RVT 1502) is a novel potent, selective, orally bioavailable glucagon receptor (GCGR) antagonist.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4309301
Biological Activity
LGD-6972 (RVT 1502) is a novel potent, selective, orally bioavailable glucagon receptor (GCGR ) antagonist; binds competitively to GCGR with high affinity and selectivity, suppressing both cAMP and glucose production in vitro.
Physicochemical Properties
M.Wt
702.9008
Formula
C43H46N2O5S
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
DMSO: ≥ 31 mg/mL
Chemical Name/SMILES
Ethanesulfonic acid, 2-[[4-[(2R)-2-[4'-(1,1-dimethylethyl)[1,1'-biphenyl]-4-yl]-3-oxo-3-[(2',4',6'-trimethyl[1,1'-biphenyl]-4-yl)amino]propyl]benzoyl]amino]-
References
1. Vajda EG, et al. Diabetes Obes Metab. 2017 Jan;19(1):24-32.
2. Vajda EG, et al. Diabetes. 2012;61(suppl 1):A252. Abstract.
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