LIT-001 trifluoroacetate | OXTR agonist

Chemical Structure : LIT-001 trifluoroacetate

CAS No.: 2245072-21-1

LIT-001 trifluoroacetate (LIT001)

Catalog No.: PC-35700Not For Human Use, Lab Use Only.

LIT-001 trifluoroacetate (LIT001) is the first nonpeptide Oxytocin receptor (OT-R) agonist with EC50 of 55 nM, Emax=96%.

Packing	Price	Stock
5 mg	$98	In stock
10 mg	$148	In stock
25 mg	$258	In stock
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Biological Activity

LIT-001 trifluoroacetate (LIT001) is the first nonpeptide Oxytocin receptor (OT-R) agonist with EC50 of 55 nM, Emax=96%.
LIT-001 efficiently relieved social interaction deficits in Oprm1−/− mice, a mouse model of autism.

Physicochemical Properties

M.Wt	645.702
Formula	C30H34F3N7O4S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-2-(Dimethylcarbamothioyl)-N-(2-methyl-4-(1-methyl1,4,5,10-tetrahydrobenzo[b]pyrazolo[3,4-e][1,4]diazepine-5- carbonyl)benzyl)pyrrolidine-1-carboxamide, trifluoroacetate

References

1. Frantz MC, et al. J Med Chem. 2018 Oct 11;61(19):8670-8692.

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LIT-001 trifluoroacetate (LIT001)

Biological Activity

Physicochemical Properties

References

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