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LPA2 antagonist 1

Chemical Structure : LPA2 antagonist 1

CAS No.: 1017606-66-4

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LPA2 antagonist 1 (LPA2-IN-1)

Catalog No.: PC-45411Not For Human Use, Lab Use Only.

LPA2 antagonist 1 is a potent, selective LPA2 (EDG4) antagonist with IC50 of 17 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

LPA2 antagonist 1 is a potent, selective LPA2 (EDG4) antagonist with IC50 of 17 nM.
LPA2 antagonist 1 inhibits the phosphorylation of Erk induced by LPA in a concentration dependent manner.
LPA2 antagonist 1 inhibits HCT-116 colon cancer cell proliferation caused by LPA in a doses dependent manner.

Physicochemical Properties

M.Wt 500.4649
Formula C20H23Cl2N5O2S2
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

Thieno[3,2-d]pyrimidin-4-amine, N-[(1S)-2-[4-[(3,4-dichlorophenyl)sulfonyl]-1-piperazinyl]-1-methylethyl]-7-methyl-

References

1. Beck HP, et al. Bioorg Med Chem Lett. 2008 Feb 1;18(3):1037-41.

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