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You are here:Home-Chemical Inhibitors & Agonists-GPCR-Free Fatty Acid Receptor (FFAR)-LY2922470
LY2922470

Chemical Structure : LY2922470

CAS No.: 1423018-12-5

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LY2922470 (LY-2922470;LY 2922470)

Catalog No.: PC-60236Not For Human Use, Lab Use Only.

LY2922470 (LY-2922470) is a potent, selective, orally available GPR40 agonist with EC50 of 7 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

LY2922470 (LY-2922470) is a potent, selective, orally available GPR40 agonist with EC50 of 7 nM.
LY2922470 displays no activity against PPARα/β/γ (>10 uM).
LY2922470 demonstrates potent, efficacious, and durable dose-dependent reductions in glucose levels along with significant increases in insulin and GLP-1 secretion in vivo.

Physicochemical Properties

M.Wt 475.603
Formula C28H29NO4S
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(S)-3-(4-((5-((8-methoxy-3,4-dihydroquinolin-1(2H)-yl)methyl)thiophen-2-yl)methoxy)phenyl)hex-4-ynoic acid

References

1. Hamdouchi C, et al. J Med Chem. 2016 Dec 22;59(24):10891-10916.

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