Lixivaptan | V2R antagonist | Probechem Biochemicals

Chemical Structure : Lixivaptan

CAS No.: 168079-32-1

Lixivaptan (VPA-985, WAY-VPA 985)

Catalog No.: PC-25955Not For Human Use, Lab Use Only.

Lixivaptan (VPA-985, WAY-VPA 985) is a potent, selective and orally active vasopressin receptor V2 (V2R) antagonist with IC50 of 1.2 and 2.3 nM for human and rat V2R, respectively.

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10 mg	$88	In stock
25 mg	$148	In stock
50 mg	$258	In stock
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Biological Activity

Lixivaptan (VPA-985, WAY-VPA 985) is a potent, selective and orally active vasopressin receptor V2 (V2R) antagonist with IC50 of 1.2 and 2.3 nM for human and rat V2R, respectively.

Physicochemical Properties

M.Wt	473.93
Formula	C27H21ClFN3O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(3-Chloro-4-(10,11-dihydro-5H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)phenyl)-5-fluoro-2-methylbenzamide

References

1. Albright JD, et al. J Med Chem. 1998 Jul 2;41(14):2442-4.

2. Chan PS, et al. Adv Exp Med Biol. 1998;449:439-43.

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Lixivaptan (VPA-985, WAY-VPA 985)

Biological Activity

Physicochemical Properties

References

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