M77976 | PDK4 inhibitor | Probechem Biochemicals

Chemical Structure : M77976

CAS No.: 394237-61-7

Catalog No.: PC-21872Not For Human Use, Lab Use Only.

M77976 is a selective inhibitor of pyruvate dehydrogenase kinase 4 (PDK4) with IC50 of 648 uM, binds to the ATP-binding pocket of PDK4.

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Biological Activity

M77976 is a selective inhibitor of pyruvate dehydrogenase kinase 4 (PDK4) with IC50 of 648 uM, binds to the ATP-binding pocket of PDK4.

M.Wt	296.33
Formula	C17H16N2O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4-(4-(4-methoxyphenyl)-5-methyl-1H-pyrazol-3-yl)benzene-1,3-diol

1. Kukimoto-Niino M, et al. Acta Crystallogr D Biol Crystallogr. 2011 Sep;67(Pt 9):763-73.

2. Wang H, et al. Cancer Metab. 2024 Jan 10;12(1):2.