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M871

Chemical Structure : M871

CAS No.: 908844-75-7

M871 (Galanin-(2-13)-Glu-His-(Pro)3-(Ala-Leu)2-Ala-amide)

Catalog No.: PC-23338Not For Human Use, Lab Use Only.

M871 (Galanin-(2-13)-Glu-His-(Pro)3-(Ala-Leu)2-Ala-amide) is a potent, selective galanin receptor type 2 (GALR2) antagonist with Ki value of 13.1 nM, >30-fold selective over GALR2.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

M871 (Galanin-(2-13)-Glu-His-(Pro)3-(Ala-Leu)2-Ala-amide) is a potent, selective galanin receptor type 2 (GALR2) antagonist with Ki value of 13.1 nM, >30-fold selective over GALR2.

Physicochemical Properties

M.Wt 2287.61
Formula C108H163N27O28
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

L-Tryptophyl-L-threonyl-L-leucyl-L-asparaginyl-L-seryl-L-alanylglycyl-L-tyrosyl-L-leucyl-L-leucylglycyl-L-prolyl-L-α-glutamyl-L-histidyl-L-prolyl-L-prolyl-L-prolyl-L-alanyl-L-leucyl-L-alanyl-L-leucyl-L-alaninamide

References

1. U. E. Sollenberg, et al. Int J Pept Res Ther. 2006;12:2965-2982.

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