MCT1-IN-4a |CAS:1448314-00-8 Probechem Biochemicals

Chemical Structure : MCT1-IN-4a

MCT1-IN-4a

Catalog No.: PC-62725Not For Human Use, Lab Use Only.

MCT1-IN-4a is a potent, selective monocarboxylate transporter 1 (MCT1) inhibitor with IC50 of 90 nM.

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Biological Activity

MCT1-IN-4a is a potent, selective monocarboxylate transporter 1 (MCT1) inhibitor with IC50 of 90 nM; exhibits significant single agent activity in MCT1 expressing GL261-luc2 syngraft model, but not in MCT4 expressing MDA-MB-231 xenograft model; has good absorption, metabolic stability, and a low drug efflux ratio.

Physicochemical Properties

M.Wt	385.419
Formula	C24H19NO4
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	7-(dibenzylamino)-2-oxo-2H-chromene-3-carboxylic acid

References

1. Gurrapu S, et al. Bioorg Med Chem Lett. 2016 Jul 15;26(14):3282-6.

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MCT1-IN-4a

Biological Activity

Physicochemical Properties

References

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