MDL-29951 | GPR17 agonist, NMDAR antagonist

Chemical Structure : MDL-29951

CAS No.: 130798-51-5

MDL-29951 (MDL 29,951, MDL29951)

Catalog No.: PC-23317Not For Human Use, Lab Use Only.

MDL-29951 (MDL-29, 951) is a potent glycine antagonist of NMDA receptor with Ki of 0.14 uM for [3H]glycine binding in vitro, also is a potent GPR17 agonist with pEC50 of 6.48.

Packing	Price	Stock
5 mg	$128	In stock
10 mg	$198	In stock
25 mg	$348	In stock
50 mg		Get quote
100 mg		Get quote

Get Quotation Now

* Please select Quantity before adding items.

or Bulk Inquiry

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Biological Activity

MDL-29951 (MDL-29, 951) is a potent glycine antagonist of NMDA receptor with Ki of 0.14 uM for [3H]glycine binding in vitro, also is a potent GPR17 agonist with pEC50 of 6.48.

Physicochemical Properties

M.Wt	302.11
Formula	C12H9Cl2NO4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-(2-Carboxyethyl)-4,6-dichloro-1H-indole-2-carboxylic acid

References

1. Baron BM, et al. J Pharmacol Exp Ther. 1992 Sep;262(3):947-56.

2. Wright SW, et al. Bioorg Med Chem Lett. 2003 Jun 16;13(12):2055-8.

3. Stephanie Hennen, et al. Sci Signal. 2013 Oct 22;6(298):ra93.

Overnight Delivery
Fast & Safe Delivery Worldwide
Rewards Program

About Us

Our Services

Site Map

Join with Us
Product Use Citations

Pharmacological Glossary Abbreviations

Abbreviations

Quality Manual

Inquiry Form
How to Order

Terms & Conditions

Credit Card Payment

Shipping Rates & Policies

Privacy Policy
sales@probechem.com

MDL-29951 (MDL 29,951, MDL29951)

Biological Activity

Physicochemical Properties

References

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

Get Quote

* Indicates a Required FieldYour information is safe with us.