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MK-2894 sodium

Chemical Structure : MK-2894 sodium

CAS No.: 1006036-88-9

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MK-2894 sodium (MK 2894 sodium;MK2894 sodium)

Catalog No.: PC-42573Not For Human Use, Lab Use Only.

MK-2894 sodium is a highly potent, selective, second generation prostaglandin E2 subtype 4 receptor (EP4) antagonist with Ki of 0.56 nM.

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25 mg $288 In stock
50 mg $458 In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

MK-2894 sodium is a highly potent, selective, second generation prostaglandin E2 subtype 4 receptor (EP4) antagonist with Ki of 0.56 nM.
MK-2894 displays >10,000-fold selectivity over EP2 receptors.
MK-2894 exhibits favorable pharmacokinetic profile and potent anti-inflammatory activity in animal models of pain/inflammation.

Physicochemical Properties

M.Wt 495.4891
Formula C25H21F3NNaO3S
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

Benzoic acid, 4-[1-[[[2,5-dimethyl-4-[[4-(trifluoromethyl)phenyl]methyl]-3-thienyl]carbonyl]amino]cyclopropyl]-, sodium salt (1:1)

References

1. Blouin M, et al. J Med Chem. 2010 Mar 11;53(5):2227-38.

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