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Chemical Structure : MK-2894 sodium
CAS No.: 1006036-88-9
Catalog No.: PC-42573Not For Human Use, Lab Use Only.
MK-2894 sodium is a highly potent, selective, second generation prostaglandin E2 subtype 4 receptor (EP4) antagonist with Ki of 0.56 nM.
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|---|---|---|---|
| 10 mg | $188 | In stock | |
| 25 mg | $288 | In stock | |
| 50 mg | $458 | In stock | |
| 100 mg | Get quote |
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MK-2894 sodium is a highly potent, selective, second generation prostaglandin E2 subtype 4 receptor (EP4) antagonist with Ki of 0.56 nM.
MK-2894 displays >10,000-fold selectivity over EP2 receptors.
MK-2894 exhibits favorable pharmacokinetic profile and potent anti-inflammatory activity in animal models of pain/inflammation.
| M.Wt | 495.4891 | |
| Formula | C25H21F3NNaO3S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
Benzoic acid, 4-[1-[[[2,5-dimethyl-4-[[4-(trifluoromethyl)phenyl]methyl]-3-thienyl]carbonyl]amino]cyclopropyl]-, sodium salt (1:1) |
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1. Blouin M, et al. J Med Chem. 2010 Mar 11;53(5):2227-38.
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