MK-571 sodium is a potent and specific LTD4 receptor antagonist with Ki of 0.22 nM.
MK-571 sodium effectively blocks LTD4 activation of recombinant human and mouse CysLT1 receptors.
MK-571 sodium also is an inhibitor of multidrug resistance protein-1 (MRP1) mediated transportorally active.
Physicochemical Properties
M.Wt
537.069
Formula
C26H26ClN2NaO3S2
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
H2O: 50 mM in H2O (26.85 mg/mL, ultrasonic needed)
