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Chemical Structure : ML301
Catalog No.: PC-20492Not For Human Use, Lab Use Only.
ML301 is a selective full (79-93%) neurotensin-1 (NTR1) receptor agonist with EC50 of 2.0-4.1 uM, good selectivity relative to NTR2 and GPR35.
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ML301 is a selective full (79-93%) neurotensin-1 (NTR1) receptor agonist with EC50 of 2.0-4.1 uM, good selectivity relative to NTR2 and GPR35.
ML301 showed good activity in a Ca mobilization FLIPR assay (93% efficacy at 298 nM), consistent with it functioning via the Gq coupled pathway.
| M.Wt | 522.99 | |
| Formula | C27H27ClN4O5 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Hershberger PM, et al. Bioorg Med Chem Lett. 2014 Jan 1;24(1):262-7.
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