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MPX-007

Chemical Structure : MPX-007

CAS No.: 1688685-29-1

MPX-007 (MPX007)

Catalog No.: PC-22451Not For Human Use, Lab Use Only.

MPX-007 is a selective GluN2A antagonist, inhibits GluN2A-containing NMDA receptors expressed in HEK cells with IC50 of 27 nM.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

MPX-007 is a selective GluN2A antagonist, inhibits GluN2A-containing NMDA receptors expressed in HEK cells with IC50 of 27 nM.

Physicochemical Properties

M.Wt 453.48
Formula C18H17F2N5O3S2
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

2-Pyrazinecarboxamide, 5-[[[(3,4-difluorophenyl)sulfonyl]amino]methyl]-6-methyl-N-[(2-methyl-5-thiazolyl)methyl]-

References

1. Jiang L, et al. Acta Pharm Sin B. 2024 May;14(5):1987-2005.

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