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Chemical Structure : MRGPRX2 antagonist C9
CAS No.: 1274013-03-4
Catalog No.: PC-38068Not For Human Use, Lab Use Only.
MRGPRX2 antagonist C9 is a potent and selective MRGPRX2 inverse agonist (antagonist) with Ki of 43 nM.
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MRGPRX2 antagonist C9 is a potent and selective MRGPRX2 inverse agonist (antagonist) with Ki of 43 nM.
MRGPRX2 antagonist C9 displays no antagonist activity towards NK1R or MRGPRX4.
MRGPRX2 antagonist C9 inhibits (R)-ZINC-3573-stimulated LAD2 human mast cell degranulation in a concentration-dependent manner.
| M.Wt | 275.344 | |
| Formula | C12H9N3OS2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
3-(thiazol-2-ylmethyl)-2-thioxo-2,3-dihydroquinazolin-4(1H)-one |
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1. Can Cao, et al. Nature. 2021 Dec;600(7887):170-175.
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