MRGPRX2 antagonist C9 |CAS:1274013-03-4 Probechem Biochemicals

Chemical Structure : MRGPRX2 antagonist C9

CAS No.: 1274013-03-4

MRGPRX2 antagonist C9 (ZINC49534341)

Catalog No.: PC-38068Not For Human Use, Lab Use Only.

MRGPRX2 antagonist C9 is a potent and selective MRGPRX2 inverse agonist (antagonist) with Ki of 43 nM.

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Biological Activity

MRGPRX2 antagonist C9 is a potent and selective MRGPRX2 inverse agonist (antagonist) with Ki of 43 nM.
MRGPRX2 antagonist C9 displays no antagonist activity towards NK1R or MRGPRX4.
MRGPRX2 antagonist C9 inhibits (R)-ZINC-3573-stimulated LAD2 human mast cell degranulation in a concentration-dependent manner.

Physicochemical Properties

M.Wt	275.344
Formula	C12H9N3OS2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-(thiazol-2-ylmethyl)-2-thioxo-2,3-dihydroquinazolin-4(1H)-one

References

1. Can Cao, et al. Nature. 2021 Dec;600(7887):170-175.

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MRGPRX2 antagonist C9 (ZINC49534341)

Biological Activity

Physicochemical Properties

References

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