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Chemical Structure : MRS7292
Catalog No.: PC-22973Not For Human Use, Lab Use Only.
MRS7292 is an allosteric, non-competitive inhibitor of human dopamine transporter (DAT) with EC50 of 35 nM, and norepinephrine transporter (NET), also is a potent A3AR agonist with Ki of 5.38 nM.
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MRS7292 is an allosteric, non-competitive inhibitor of human dopamine transporter (DAT) with EC50 of 35 nM, and norepinephrine transporter (NET), also is a potent A3AR agonist with Ki of 5.38 nM.
| M.Wt | 459.91 | |
| Formula | C20H18ClN5O4S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Tosh DK, et al. J Med Chem. 2017 Apr 13;60(7):3109-3123.
2. Srivastava DK, et al. Nature. 2024 Aug;632(8025):672-677.
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