MRS8209

Chemical Structure : MRS8209

Catalog No.: PC-23512Not For Human Use, Lab Use Only.

MRS8209 is a potent, peripheral subtype-selective 5-HT2B serotonin receptor antagonist with Ki of 4.27 nM (human 5-HT2B), shows reduced affinity at the m5-HT2BR and r5-HT2BR (100-fold and 10-fold).

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Biological Activity

MRS8209 is a potent, peripheral subtype-selective 5-HT2B serotonin receptor antagonist with Ki of 4.27 nM (human 5-HT2B), shows reduced affinity at the m5-HT2BR and r5-HT2BR (100-fold and 10-fold).

Physicochemical Properties

M.Wt	466.28
Formula	C17H19IN6O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(1R,2R,3S,4R,5S)-4-(6-(Cyclopentylamino)-2-iodo-9H-purin-9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carbonitrile

References

1. Tosh DK, et al. J Med Chem. 2024 Nov 26. doi: 10.1021/acs.jmedchem.4c02174.

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MRS8209

Biological Activity

Physicochemical Properties

References

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