You are here:Home-Chemical Inhibitors & Agonists-GPCR-Proton-sensing GPCRs-MS48107
MS48107

Chemical Structure : MS48107

CAS No.: 2375070-79-2

MS48107 (MS 48107)

Catalog No.: PC-72990Not For Human Use, Lab Use Only.

MS48107 (MS 48107) is a potent, selective, positive allosteric modulator of G protein-coupled receptor 68 (GPR68, Log(αβ/KB)=6.83).

Packing Price Stock Quantity
10 mg $148 In stock
25 mg $268 In stock
50 mg $428 In stock
100 mg Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

MS48107 (MS 48107) is a potent, selective, positive allosteric modulator of G protein-coupled receptor 68 (GPR68, Log(αβ/KB)=6.83).
MS48107 displays good selectivity against all human GPCRome in PRESTO-Tango screening assays.
MS48107 was bioavailable and brain-penetrant in mice.

Physicochemical Properties

M.Wt 417.444
Formula C23H20FN5O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

(2-(4-Amino-6-((4-phenoxybenzyl)amino)-1,3,5-triazin-2-yl)-3-fluorophenyl)methanol

References

1. Xufen Yu, et al. J Med Chem. 2019 Aug 22;62(16):7557-7574.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: