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Macimorelin

Chemical Structure : Macimorelin

CAS No.: 381231-18-1

Macimorelin (JMV-1843, EP-1572, AEZS-130)

Catalog No.: PC-23038Not For Human Use, Lab Use Only.

Macimorelin (JMV-1843, EP-1572) is a GH secretagogue and orally active GHSR agonist with binding IC50 of 22.9 nM to cloned human GHS−R 1a receptor.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Macimorelin (JMV-1843, EP-1572) is a GH secretagogue and orally active GHSR agonist with binding IC50 of 22.9 nM to cloned human GHS−R 1a receptor.

Physicochemical Properties

M.Wt 474.57
Formula C26H30N6O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

2-Methylalanyl-N-[(1R)-1-(formylamino)-2-(1H-indol-3-yl)ethyl]-D-tryptophanamide

References

1. Guerlavais V, et al. J Med Chem. 2003. PMID: 12646029

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