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Milveterol

Chemical Structure : Milveterol

CAS No.: 652990-07-3

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Milveterol (GSK 159797)

Catalog No.: PC-62004Not For Human Use, Lab Use Only.

Milveterol (GSK 159797) is a potent, selective long-acting β2 adrenoceptor agonist with pEC50 of 10.2 in cell-based assays, displays good β2/β1 selectivity (>300-fold).

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    Milveterol (GSK 159797) is a potent, selective long-acting β2 adrenoceptor agonist with pEC50 of 10.2 in cell-based assays, displays good β2/β1 selectivity (>300-fold).
    Milveterol (GSK 159797) demonstrates high potency in vitro and long duration of action in a guinea pig model of bronchoprotection.

    Physicochemical Properties

    M.Wt 435.524
    Formula C25H29N3O4
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    N-(2-hydroxy-5-((R)-1-hydroxy-2-((4-(((R)-2-hydroxy-2-phenylethyl)amino)phenethyl)amino)ethyl)phenyl)formamide

    References

    1. Jacobsen JR, et al. Bioorg Med Chem Lett. 2012 Jan 15;22(2):1213-8.

    2. Fuso L, et al. Curr Med Chem. 2013;20(12):1477-95.

    3. Jacobsen JR, et al. Bioorg Med Chem Lett. 2014 Jun 15;24(12):2625-30.

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