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Chemical Structure : Mozavaptan
CAS No.: 137975-06-5
Catalog No.: PC-45459Not For Human Use, Lab Use Only.
Mozavaptan (OPC-31260) is a potent, selective nonpeptide vasopressin V2 receptor antagonist with IC50 of 14 nM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 50 mg | $98 | In stock | |
| 100 mg | $158 | In stock | |
| 250 mg | $258 | In stock | |
| 1 g | Get quote |
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Mozavaptan (OPC-31260) is a potent, selective nonpeptide vasopressin V2 receptor antagonist with IC50 of 14 nM.
Mozavaptan 100-fold less potent for VP1 (IC50=1.2 uM).
Mozavaptan dose-dependently increases urine flow and decreases urine osmolality in normal conscious rats; orally effective.
| M.Wt | 427.5381 | |
| Formula | C27H29N3O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: 6.2 mg/mL (Need warming) |
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| Chemical Name/SMILES |
Benzamide, N-[4-[[5-(dimethylamino)-2,3,4,5-tetrahydro-1H-1-benzazepin-1-yl]carbonyl]phenyl]-2-methyl- |
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1. Yamamura Y, et al. Br J Pharmacol. 1992 Apr;105(4):787-91.
2. Tsuboi Y, et al. J Endocrinol. 1994 Nov;143(2):227-34.
3. Wang X, et al. J Am Soc Nephrol. 2005 Apr;16(4):846-51.
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