N-desmethyl Enzalutamide |CAS:1242137-16-1 Probechem Biochemicals

Chemical Structure : N-desmethyl Enzalutamide

CAS No.: 1242137-16-1

Catalog No.: PC-45933Not For Human Use, Lab Use Only.

Amajor metabolite of Enzalutamide (MDV3100) which is an androgen-receptor (AR) antagonist for treatment of prostate cancer..

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50 mg	$520	In stock
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Biological Activity

Amajor metabolite of Enzalutamide (MDV3100) which is an androgen-receptor (AR) antagonist for treatment of prostate cancer.

M.Wt	450.4094
Formula	C20H14F4N4O2S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	DMSO: ≥ 48 mg/mL
Chemical Name/SMILES	Benzamide, 4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-thioxo-1-imidazolidinyl]-2-fluoro-

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2. Richards J, et al. Cancer Res. 2012 May 1;72(9):2176-82.

3. Gibbons JA, et al. Clin Pharmacokinet. 2015 Oct;54(10):1043-55.