N-desmethyl Enzalutamide |CAS:1242137-16-1 Probechem Biochemicals

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Chemical Structure : N-desmethyl Enzalutamide

CAS No.: 1242137-16-1

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N-desmethyl Enzalutamide (N-desmethyl MDV3100, N-desmethyl MDV-3100)

Catalog No.: PC-45933Not For Human Use, Lab Use Only.

N-desmethyl Enzalutamide is a major metabolite of Enzalutamide (MDV3100) which is an androgen-receptor (AR) antagonist for treatment of prostate cancer.

Packing	Price	Stock
10 mg	$78	In stock
25 mg	$128	In stock
50 mg	$198	In stock
100 mg		Get quote

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

N-desmethyl Enzalutamide is a major metabolite of Enzalutamide (MDV3100) which is an androgen-receptor (AR) antagonist for treatment of prostate cancer.

Physicochemical Properties

M.Wt	450.4094
Formula	C20H14F4N4O2S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	DMSO: ≥ 48 mg/mL
Chemical Name/SMILES	Benzamide, 4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-thioxo-1-imidazolidinyl]-2-fluoro-

References

1. Tran C, et al. Science. 2009 May 8;324(5928):787-90.

2. Richards J, et al. Cancer Res. 2012 May 1;72(9):2176-82.

3. Gibbons JA, et al. Clin Pharmacokinet. 2015 Oct;54(10):1043-55.

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N-desmethyl Enzalutamide (N-desmethyl MDV3100, N-desmethyl MDV-3100)

Biological Activity

Physicochemical Properties

References

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