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You are here:Home-Chemical Inhibitors & Agonists-Membrane Transporter/Ion Channel-Glutamate Transporter-NA-014
NA-014

Chemical Structure : NA-014

CAS No.: 3041127-59-4

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NA-014 (NA014)

Catalog No.: PC-28283Not For Human Use, Lab Use Only.

NA-014 is a potent, selective positive allosteric modulator (PAM) of excitatory amino acid transporter 2 (EAAT2, rodent homologue glutamate transporter-1, GLT-1) with EC50 of 3.0 nM, is inactive against EAAT1 and EAAT3.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

NA-014 is a potent, selective positive allosteric modulator (PAM) of excitatory amino acid transporter 2 (EAAT2, rodent homologue glutamate transporter-1, GLT-1) with EC50 of 3.0 nM, is inactive against EAAT1 and EAAT3.

Physicochemical Properties

M.Wt 380.46
Formula C22H25FN4O
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-(4-Cyanophenyl)-N-(4-fluorophenethyl)-2-(4-methylpiperazin-1-yl)acetamide

References

1. Fontana ACK, et al. J Med Chem. 2024 Apr 25;67(8):6119-6143.

2. Reeb KL, et al. Eur J Pharmacol. 2024 Dec 5;984:177017.

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