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Chemical Structure : NTRC-824
Catalog No.: PC-22266Not For Human Use, Lab Use Only.
NTRC-824 is the first nonpeptide, selective antagonist of neurotensin receptor type 2 (NTS2/NTSR2) with IC50 of 32 nM in FLIPR assays, binding Ki of 202 nM.
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NTRC-824 is the first nonpeptide, selective antagonist of neurotensin receptor type 2 (NTS2/NTSR2) with IC50 of 32 nM in FLIPR assays, binding Ki of 202 nM.
NTRC-824 displays no significant affinity for NTS1 (Ki>30 uM).
| M.Wt | 553.55 | |
| Formula | C25H26F3N3O6S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Thomas JB, et al. J Med Chem. 2014 Sep 11;57(17):7472-7.
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