NTSR1 agonist RTI-3a

Chemical Structure : NTSR1 agonist RTI-3a

Catalog No.: PC-28389Not For Human Use, Lab Use Only.

NTSR1 agonist RTI-3a is a potent, selective partial agonist of neurotensin receptor 1 (NTSR1) with EC50 of 67 nM and Emax of 54%.

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Biological Activity

NTSR1 agonist RTI-3a is a potent, selective partial agonist of neurotensin receptor 1 (NTSR1) with EC50 of 67 nM and Emax of 54%.

M.Wt	522.99
Formula	C27H27ClN4O5
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(1-(7-chloroquinolin-4-yl)-5-(2,6-dimethoxyphenyl)-1H-pyrazole-3-carbonyl)-L-leucine

1. James B Thomas, et al. Bioorg Med Chem Lett. 2009 Mar 1;19(5):1438-41.