Netupitant | NK1R antagonist | Probechem Biochemicals

Chemical Structure : Netupitant

CAS No.: 290297-26-6

Netupitant (CID 6451149)

Catalog No.: PC-27027Not For Human Use, Lab Use Only.

Netupitant (CID 6451149) is a highly potent, selective and orally active neurokinin-1 receptor (NK1R) antagonist with Ki of 0.95 nM for hNK1 receptor, >1000-fold selective over NK2R and NK3R.

Packing	Price	Stock
25 mg	$78	In stock
50 mg	$118	In stock
100 mg	$188	In stock
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Biological Activity

Netupitant (CID 6451149) is a highly potent, selective and orally active neurokinin-1 receptor (NK1R) antagonist with Ki of 0.95 nM for hNK1 receptor, >1000-fold selective over NK2R and NK3R.

Physicochemical Properties

M.Wt	578.60
Formula	C30H32F6N4O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-(3,5-Bis(trifluoromethyl)phenyl)-N,2-dimethyl-N-(6-(4-methylpiperazin-1-yl)-4-(o-tolyl)pyridin-3-yl)propanamide

References

1. Hoffmann T, et al. Bioorg Med Chem Lett. 2006 Mar 1;16(5):1362-5.

2. Rizzi A, et al. Peptides. 2012 Sep;37(1):86-97.

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Netupitant (CID 6451149)

Biological Activity

Physicochemical Properties

References

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