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Chemical Structure : ORM-15341
CAS No.: 1297537-33-7
Catalog No.: PC-45612Not For Human Use, Lab Use Only.
The active main metabolite of ODM-201, a potent wt/mutant androgen receptor (AR) inhibitor.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $400 | In stock | |
| 50 mg | $1200 | In stock | |
| 100 mg | $1680 | In stock |
Bulk size, bulk discount!
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The active main metabolite of ODM-201, a potent wt/mutant androgen receptor (AR) inhibitor; inhibits wtAR/AR(F876L) with IC50s of 25/51 nM respectively; suppresses androgen-induced cell proliferation more efficaciously than enzalutamide or ARN-509.
| M.Wt | 396.8303 | |
| Formula | C19H17ClN6O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: ≥ 37 mg/mL |
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| Chemical Name/SMILES |
1H-Pyrazole-3-carboxamide, 5-acetyl-N-[(1S)-2-[3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-yl]-1-methylethyl]- |
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1. Moilanen AM, et al. Sci Rep. 2015 Jul 3;5:12007.
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