Chemical Structure : OSI-930
CAS No.:
728033-96-3
OSI-930
(OSI 930;OSI930)
Catalog No. : PC-42449Not For Human Use, Lab Use Only.
A potent, orally active, dual inhibitor of c-Kit and VEGFR-2 (KDR) with IC50 of 15 nM and 9 nM, respectively.
Packing Price Stock Quantity 10 mg $118 In stock 0 1 2 3 4 5 25 mg $198 In stock 0 1 2 3 4 5 50 mg $298 In stock 0 1 2 3 4 5 100 mg Get quote 0 1 2 3 4 5
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4244901
Biological Activity
OSI-930 is a potent, orally active, dual inhibitor of c-Kit and VEGFR-2 (KDR) with IC50 of 15 nM and 9 nM, respectively.
Physicochemical Properties
M.Wt
443.4416
Formula
C22H16F3N3O2S
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
2-Thiophenecarboxamide, 3-[(4-quinolinylmethyl)amino]-N-[4-(trifluoromethoxy)phenyl]-
References
1. Garton AJ, et al. Cancer Res.
2. Yap TA, et al. Clin Cancer Res.
3. Patel JP, et al. Bioorg Med Chem Lett.
4. Macpherson IR, et al. Eur J Cancer.
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