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Chemical Structure : Obicetrapib
CAS No.: 866399-87-3
Catalog No.: PC-63559Not For Human Use, Lab Use Only.
Obicetrapib (AMG899, TA-8995, DEZ-001) is a potent, selective and orally active cholesteryl ester transfer protein (CETP) inhibitor for treatment of dyslipidaemia.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $258 | In stock | |
| 10 mg | $398 | In stock | |
| 25 mg | $598 | In stock | |
| 50 mg | Get quote | ||
| 100 mg | Get quote |
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Obicetrapib (AMG899, TA-8995, DEZ-001) is a potent, selective and orally active cholesteryl ester transfer protein (CETP) inhibitor for treatment of dyslipidaemia.
| M.Wt | 722.609 | |
| Formula | C32H31F9N4O5 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
4-[2-[[3,5-bis(trifluoromethyl)phenyl]methyl-[(2R,4S)-1-ethoxycarbonyl-2-ethyl-6-(trifluoromethyl)-3,4-dihydro-2H-quinolin-4-yl]amino]pyrimidin-5-yl]oxybutanoic acid |
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1. Ford J, et al. Br J Clin Pharmacol. 2014 Sep;78(3):498-508.
2. Hovingh GK, et al. Lancet. 2015 Aug 1;386(9992):452-60.
3, Nicholls SJ, et al. Nat Med. 2022 Aug;28(8):1672-1678.
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