Obicetrapib (AMG899, TA-8995) | CETP inhibitor

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Chemical Structure : Obicetrapib

CAS No.: 866399-87-3

Obicetrapib (AMG-899, AMG899, TA-8995, DEZ-001)

Catalog No.: PC-63559Not For Human Use, Lab Use Only.

Obicetrapib (AMG899, TA-8995, DEZ-001) is a potent, selective and orally active cholesteryl ester transfer protein (CETP) inhibitor for treatment of dyslipidaemia.

Packing	Price	Stock
5 mg	$258	In stock
10 mg	$398	In stock
25 mg	$598	In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Obicetrapib (AMG899, TA-8995, DEZ-001) is a potent, selective and orally active cholesteryl ester transfer protein (CETP) inhibitor for treatment of dyslipidaemia.

Physicochemical Properties

M.Wt	722.609
Formula	C32H31F9N4O5
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	4-[2-[[3,5-bis(trifluoromethyl)phenyl]methyl-[(2R,4S)-1-ethoxycarbonyl-2-ethyl-6-(trifluoromethyl)-3,4-dihydro-2H-quinolin-4-yl]amino]pyrimidin-5-yl]oxybutanoic acid

References

1. Ford J, et al. Br J Clin Pharmacol. 2014 Sep;78(3):498-508.
2. Hovingh GK, et al. Lancet. 2015 Aug 1;386(9992):452-60.
3, Nicholls SJ, et al. Nat Med. 2022 Aug;28(8):1672-1678.

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Obicetrapib (AMG-899, AMG899, TA-8995, DEZ-001)

Biological Activity

Physicochemical Properties

References

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