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Obicetrapib

Chemical Structure : Obicetrapib

CAS No.: 866399-87-3

Obicetrapib (AMG-899;AMG899;TA-8995;DEX-001)

Catalog No.: PC-63559Not For Human Use, Lab Use Only.

Obicetrapib (AMG-899, TA-8995, DEX-001) is a potent, selective and orally active cholesteryl ester transfer protein (CETP) inhibitor for treatment of dyslipidaemia.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Obicetrapib (AMG-899, TA-8995, DEX-001) is a potent, selective and orally active cholesteryl ester transfer protein (CETP) inhibitor for treatment of dyslipidaemia.

Physicochemical Properties

M.Wt 722.609
Formula C32H31F9N4O5
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

4-[2-[[3,5-bis(trifluoromethyl)phenyl]methyl-[(2R,4S)-1-ethoxycarbonyl-2-ethyl-6-(trifluoromethyl)-3,4-dihydro-2H-quinolin-4-yl]amino]pyrimidin-5-yl]oxybutanoic acid

References

1. Ford J, et al. Br J Clin Pharmacol. 2014 Sep;78(3):498-508.
2. Hovingh GK, et al. Lancet. 2015 Aug 1;386(9992):452-60.
3, Nicholls SJ, et al. Nat Med. 2022 Aug;28(8):1672-1678.

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