Chemical Structure : Omapatrilat
CAS No.:
167305-00-2
Omapatrilat
(BMS-186716, BMS186716)
Catalog No. : PC-45435Not For Human Use, Lab Use Only.
Omapatrilat (BMS-186716) is a potent, dual inhibitor of the metalloproteases ACE and NEP with Ki of 0.64 nM and 0.45 nM, respectively.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4543501
Biological Activity
Omapatrilat (BMS-186716) is a potent, dual inhibitor of the metalloproteases ACE and NEP with Ki of 0.64 nM and 0.45 nM, respectively.
Physicochemical Properties
M.Wt
408.5349
Formula
C19H24N2O4S2
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
DMSO: ≥ 31 mg/mL
Chemical Name/SMILES
7H-Pyrido[2,1-b][1,3]thiazepine-7-carboxylic acid, octahydro-4-[[(2S)-2-mercapto-1-oxo-3-phenylpropyl]amino]-5-oxo-, (4S,7S,10aS)-
References
1. Robl JA, et al. J Med Chem.
2. Fryer RM, et al. Br J Pharmacol.
3. Burrell LM, et al. Am J Hypertens
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