Chemical Structure : Org 25543
CAS No.:
495076-64-7
Org 25543
(Org-25543;Org25543)
Catalog No.: PC-60445Not For Human Use, Lab Use Only.
Org 25543 is a potent, highly selective glycine transporter 1 (GlyT2) inhibitor with IC50 of 16 nM with negligible affinity for GlyT1.
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| 10 mg | $368 | In stock | |
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Purity & Documentation Purity:
>98% (HPLC)
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Biological Activity
Org 25543 is a potent, highly selective glycine transporter 1 (GlyT2) inhibitor with IC50 of 16 nM with negligible affinity for GlyT1.
Physicochemical Properties
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M.Wt
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448.988
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Formula
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C24H33ClN2O4
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Appearance
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Solid
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CAS No.
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Storage
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- Solide Powder
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-20 °C 12 Months; 4°C 6 Months
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- In Solvent
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-80 °C 6 Months; -20°C 6 Months
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Shipping
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Solubility
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10 mM in DMSO
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Chemical Name/SMILES
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Benzamide, N-[[1-(dimethylamino)cyclopentyl]methyl]-3,5-dimethoxy-4-(phenylmethoxy)-, monohydrochloride (9CI)
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References
1. Morita K, et al. J Pharmacol Exp Ther. 2008 Aug;326(2):633-45.
2. Rousseau F, et al. J Neurosci. 2008 Sep 24;28(39):9755-68.
3. Romei C, et al. J Neurochem. 2011 Oct;119(1):50-63.
4. Mingorance-Le Meur A, et al. Br J Pharmacol. 2013 Nov;170(5):1053-63.
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