P-retigabine | Kv7 activator | Probechem Biochemicals

Chemical Structure : P-retigabine

P-retigabine (P-RTG)

Catalog No.: PC-27792Not For Human Use, Lab Use Only.

P-retigabine (P-RTG) is a Retigabine analog with improved brain distribution and neuronal Kv7 channel activator with EC50 of 2.04 uM (KCNQ2, Kv7.2), displays moderate anticonvulsant efficacy.

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Biological Activity

P-retigabine (P-RTG) is a Retigabine analog with improved brain distribution and neuronal Kv7 channel activator with EC50 of 2.04 uM (KCNQ2, Kv7.2), displays moderate anticonvulsant efficacy.

Physicochemical Properties

M.Wt	341.39
Formula	C19H20FN3O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	ethyl N-[2-amino-4-((4-fluorobenzyl)(prop-2-ynyl)amino)phenyl]carbamate

References

1. Yang-Ming Zhang, et al. J Med Chem. 2021 May 13;64(9):5816-5837.

2. Zhou P, et al. Mol Pharmacol. 2015 Jan;87(1):31-8.

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P-retigabine (P-RTG)

Biological Activity

Physicochemical Properties

References

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