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PDE1-IN-2

Chemical Structure : PDE1-IN-2

CAS No.: 1904611-63-7

PDE1-IN-2 (PDE1C inhibitor)

Catalog No.: PC-42399Not For Human Use, Lab Use Only.

PDE1-IN-2 is a potent, selective PDE1C inhibitor with IC50 of 6 nM, weakly inhibits PDE1B and PDE1A with IC50 of 140 and 164 nM, respectvely.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

PDE1-IN-2 is a potent, selective PDE1C inhibitor with IC50 of 6 nM, weakly inhibits PDE1B and PDE1A with IC50 of 140 and 164 nM, respectvely.

Physicochemical Properties

M.Wt 381.26754
Formula C16H21BrN4O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

DMSO: 10 mM

Chemical Name/SMILES

1,2,4-Triazolo[4,3-a]pyrazin-8(7H)-one, 6-bromo-7-(cyclopentylmethyl)-3-(tetrahydro-2H-pyran-4-yl)-

References

1. Patent WO2016055618A1, compound Example 36.

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