PDE10A-IN-31 |CAS:1639889-98-7 Probechem Biochemicals

Chemical Structure : PDE10A-IN-31

PDE10A-IN-31 (PDE10A inhibitor 31)

Catalog No.: PC-62737Not For Human Use, Lab Use Only.

PDE10A-IN-31 is a potent, highly selective PDE10A inhibitor with IC50 of 2 nM for both rPDE10A and hPDE10A.

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Biological Activity

PDE10A-IN-31 is a potent, highly selective PDE10A inhibitor with IC50 of 2 nM for both rPDE10A and hPDE10A.
PDE10A-IN-31 dispalys >2,000-fold selective over PDE1B/2A/3B/4D/5A/7A9A, weak activity on CYP isoforms.
PDE10A-IN-31 displays excellent pharmacokinetic properties.

Physicochemical Properties

M.Wt	477.524
Formula	C28H23N5O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(E)-4-(8-morpholino-2-(2-(quinolin-2-yl)vinyl)imidazo[1,2-b]pyridazin-3-yl)benzoic acid

References

1. Meegalla SK, et al. Bioorg Med Chem Lett. 2016 Sep 1;26(17):4216-22.

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PDE10A-IN-31 (PDE10A inhibitor 31)

Biological Activity

Physicochemical Properties

References

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