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You are here:Home-Chemical Inhibitors & Agonists-Membrane Transporter/Ion Channel-Microsomal Triglyceride Transfer Protein (MTP)-PF-02575799
PF-02575799

Chemical Structure : PF-02575799

CAS No.: 863491-70-7

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PF-02575799 (PF02575799)

Catalog No.: PC-63288Not For Human Use, Lab Use Only.

PF-02575799 is a highly potent microsomal triglyceride transfer protein (MTP) inhibitor with IC50 of 0.77 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    PF-02575799 is a highly potent microsomal triglyceride transfer protein (MTP) inhibitor with IC50 of 0.77 nM.
    PF-02575799 produces appreciable triglyceride effects at its minimally effective dose (10 mg/kg), significantly increases alanine transaminase at 100 mg/kg.

    Physicochemical Properties

    M.Wt 680.78
    Formula C42H37FN4O4
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    N-[(1S)-2-[[(4-Fluorophenyl)methyl]methylamino]-2-oxo-1-phenylethyl]-2-[[[4'-(1-methylethoxy)[1,1'-biphenyl]-2-yl]carbonyl]amino]-6-quinolinecarboxamide

    References

    1. Robinson RP, et al. Bioorg Med Chem Lett. 2011 Jul 15;21(14):4150-4.

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