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Chemical Structure : PF-03246799
Catalog No.: PC-61081Not For Human Use, Lab Use Only.
PF-03246799 (PF-3246799) is a potent and selective 5-HT2C receptor agonist with EC50 of 190 nM, with excellent selectivity for 5-HT2C over 5-HT2A.
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PF-03246799 (PF-3246799) is a potent and selective 5-HT2C receptor agonist with EC50 of 190 nM, with excellent selectivity for 5-HT2C over 5-HT2A.
PF-03246799 (PF-3246799) has minimal activation at either the 5-HT(2A) or 5-HT(2B) receptors.
PF-03246799 (PF-3246799)demonstrates robust efficacy in preclinical canine model of stress urinary incontinence (SUI) and attractive pharmacokinetic and safety properties.
| M.Wt | 239.322 | |
| Formula | C15H17N3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Andrews MD, et al. Bioorg Med Chem Lett. 2011 May 1;21(9):2715-20.
2. Dvorak CA, et al. ACS Med Chem Lett. 2015 Jul 20;6(9):1015-8.
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