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PF-03382792

Chemical Structure : PF-03382792

CAS No.: 1400811-63-3

PF-03382792 (PF-3382792)

Catalog No.: PC-61883Not For Human Use, Lab Use Only.

PF-03382792 is a potent, brain penetrant 5-HT4 partial agonist with Ki of 2.7 nM and an EC50 of 0.9 nM for 5-HT4d, produces moderate increases in cortical Ach in the rat prefrontal cortex.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    PF-03382792 is a potent, brain penetrant 5-HT4 partial agonist with Ki of 2.7 nM and an EC50 of 0.9 nM for 5-HT4d, produces moderate increases in cortical Ach in the rat prefrontal cortex.

    Physicochemical Properties

    M.Wt 433.52
    Formula C23H32FN3O4
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    1H-Indole-1-carboxamide, 6-fluoro-2,3-dihydro-3,3-dimethyl-2-oxo-N-((1-((tetrahydro-4-hydroxy-2H-pyran-4-yl)methyl)-4-piperidinyl)methyl)-

    References

    1. Michael A Brodney, et al. J Med Chem. 2012 Nov 8;55(21):9240-54.

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