PF-03382792 | 5-HT4 agonist | Probechem Biochemicals

Chemical Structure : PF-03382792

PF-03382792 (PF-3382792)

Catalog No.: PC-61883Not For Human Use, Lab Use Only.

PF-03382792 is a potent, brain penetrant 5-HT4 partial agonist with Ki of 2.7 nM and an EC50 of 0.9 nM for 5-HT4d, produces moderate increases in cortical Ach in the rat prefrontal cortex.

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Biological Activity

PF-03382792 is a potent, brain penetrant 5-HT4 partial agonist with Ki of 2.7 nM and an EC50 of 0.9 nM for 5-HT4d, produces moderate increases in cortical Ach in the rat prefrontal cortex.

Physicochemical Properties

M.Wt	433.52
Formula	C23H32FN3O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	1H-Indole-1-carboxamide, 6-fluoro-2,3-dihydro-3,3-dimethyl-2-oxo-N-((1-((tetrahydro-4-hydroxy-2H-pyran-4-yl)methyl)-4-piperidinyl)methyl)-

References

1. Michael A Brodney, et al. J Med Chem. 2012 Nov 8;55(21):9240-54.

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PF-03382792 (PF-3382792)

Biological Activity

Physicochemical Properties

References

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